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Puas yog los ntawm inhibition ntawm acetylcholinesterase?

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Puas yog los ntawm inhibition ntawm acetylcholinesterase?
Puas yog los ntawm inhibition ntawm acetylcholinesterase?

Video: Puas yog los ntawm inhibition ntawm acetylcholinesterase?

Video: Puas yog los ntawm inhibition ntawm acetylcholinesterase?
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Lub enzyme inactivation, induced los ntawm ntau yam inhibitors, ua rau acetylcholine tsub zuj zuj, hyperstimulation ntawm nicotinic thiab muscarinic receptors, thiab cuam tshuam neurotransmission. Yog li, acetylcholinesterase inhibitors, cuam tshuam nrog cov enzyme raws li lawv lub hom phiaj tseem ceeb, tau siv los ua cov tshuaj cuam tshuam thiab co toxins.

Yuav ua li cas thaum koj inhibit acetylcholinesterase?

Acetylcholinesterase inhibitors (AChEIs) feem ntau hu ua cholinesterase inhibitors, inhibits enzyme acetylcholinesterase los ntawm kev rhuav tshem cov neurotransmitter acetylcholine rau hauv choline thiab acetate, yog li nce qib thiab sijhawm ua haujlwm. ntawm acetylcholine nyob rau hauv lub hauv paus paj hlwb, autonomic…

Qhov tshwm sim ntawm acetylcholinesterase yog dab tsi?

Nws tam sim ntawd tawg lossis hydrolyzes acetylcholine (ACh), ib txwm tshwm sim neurotransmitter, rau hauv acetic acid thiab choline. [1] Lub luag haujlwm tseem ceeb ntawm AChE yog txhawm rau txiav tawm cov kab mob neuronal thiab kev taw qhia ntawm synapses los tiv thaiv ACh dispersal thiab ua kom cov neeg nyob ze

Acetylcholinesterase inhibitor siv rau dab tsi?

Kev siv lub ntsiab ntawm cholinesterase inhibitors yog rau kho dementia hauv cov neeg mob Alzheimer's diseaseCov neeg mob Alzheimer's tau txo qis ntawm acetylcholine hauv lub hlwb. Cholinesterase inhibitors tau pom tias muaj kev cuam tshuam me me rau cov tsos mob dementia xws li kev paub.

Cov piv txwv ntawm acetylcholinesterase inhibitors yog dab tsi?

Acetylcholinesterase Inhibitors, Central

  • Txhob Cia Siab.
  • Aricept.
  • Aricept ODT.
  • donepezil.
  • Ydonepezil transdermal.
  • Exelon.
  • Exelon Patch.
  • galantamine.

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